Found 128 of ki for VOLTAGE-DEPENDENT L-TYPE CALCIUM CHANNEL SUBUNIT ALPHA-1S
having polymerids = 50000969,50002691 and
complexids = 50000903,50024737,50000735
having polymerids = 50000969,50002691 and
complexids = 50000903,50024737,50000735
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]nitrendipine from calcium channel receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.205nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel from rat brain cortex homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Inhibitory constant against calcium channel receptors (CCRs) from rat cortex homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.499nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel from rat brain cortex homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel from rat brain cortex homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel from rat brain cortex homogenateMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rattus norvegicus)
Prestwick Chemical
Curated by ChEMBL
Prestwick Chemical
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Invitro evaluation against RXR-alpha in CV-1 cells by cotransfection assay was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel from rat brain cortex homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Displacement of [3H]nitrendipine from calcium channel receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel from rat brain cortex homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel from rat brain cortex homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]nitrendipine from calcium channel receptorMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibitory constant against calcium channel receptors (CCRs)More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]nitrendipine from calcium channel receptorMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membrane.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membrane.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Displacement of [3H]-diltiazem from L-type calcium channel of guinea pig striated muscleMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel from rat brain cortex homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Displacement of [3H]nitrendipine from calcium channel receptorMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Inhibition of [3H]D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Displacement of verapamil from L-type calcium channel binding siteMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 78nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 84nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 85nMAssay Description:Displacement of [3H]-diltiazem from L-type calcium channel of guinea pig striated muscleMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Displacement of [3H]diltiazem from L-type calcium channel in Sprague-Dawley rat cardiac myocytes by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 87nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
Affinity DataKi: 99nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
Affinity DataKi: 118nMAssay Description:Displacement of [3H]nitrendipine from calcium channel receptorMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 173nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Displacement of [3H]diltiazem from L-type calcium channel in Sprague-Dawley rat cardiac myocytes by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Displacement of [3H]nitrendipine from calcium channel receptorMore data for this Ligand-Target Pair
Affinity DataKi: 217nMAssay Description:Displacement of diltiazem from L-type calcium channel binding siteMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 254nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair